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|Product Name:||Toremifene Citrate||CAS:||89778-27-8|
|Type:||Pharmaceutical Intermediate||Appearance:||White Powder|
|Application:||Pharm Intermediates||Other Name:||Arimidex|
|Product Name:||Toremifene citrate|
|Synonyms:||(z)-4-chloro-1,2-diphenyl-1-(4-(2-(n,n-dimethylamino)ethoxy)phenyl)-1-butene;2-(4-(4-chloro-1,2-diphenyl-1-butenyl)phenoxy)-n,n-dimethyl-ethanamin(z)-ethanamin;2-hydroxy-1,2,3-propanetricarboxylate(1:1);fareston;fc1157a;nk622;TOREMIFENE CITRATE;(z)-2-[4-(4-chloro-1,2-diphenyl-1-butenyl)phenoxy]-n,n-dimethyl-ethanamine 2-hydroxy-1,2,3-propanetricarboxylate|
|Product Categories:||Active Pharmaceutical Ingredients;Amines;Aromatics;Inhibitors;Intermediates & Fine Chemicals;Pharmaceuticals;XYREM;Analgesics|
Toremifene Citrate (Fareston) is an anti-estrogenic medication, a SERM officially classified as a non-steroidal triphenylethylene derivative. As an anti-estrogen, Fareston functions by binding or attaching to the estrogen receptors in various tissues throughout the body creating a competition between it and the estrogen hormone. By attaching to the varying receptors this prevents the estrogen hormone from binding and performing its intended action. Primarily this will be beneficial in that it prevents the estrogen hormone from binding to the estrogen receptors in the mammary tissue. In fact, while other SERM’s carry this ability Fareston has been shown to carry it to the strongest level making it an excellent choice for the anabolic steroid user on cycle in the fight against gynecomastia.
Aromatase inhibitors (AIs) include compounds such as Arimidex (Anastrozole), Aromasin (Exemestane), and Letrozole (Femara). Although the two fall under the category of anti-estrogens, they are both sub- categories that branch off into their own families, as SERMs and AIs differ greatly in their mechanism of action within the human body concerning how they control or block Estrogen. There has been much misunderstanding and misconception in previous decades as to what each of these do, and this should always be first clarified to the reader before describing Toremifene.
Formestane is a second generation, irreversible, steroidal aromatase inhibitor. It inhibits the aromatase enzyme responsible for converting androgens to estrogens, thereby preventing estrogen production. Breast cancer may be estrogen sensitive or insensitive. A majority of breast cancers are estrogen sensitive. Estrogen sensitive breast cancer cells depend on estrogen for viability. Thus removal of estrogen from the body can be an effective treatment for hormone sensitive breast cancers. Formestane has been targeted specifically for the treatment of postmenopausal women. Unlike premenopausal women who produce most estrogen in the ovaries, postmenopausal women produce most estrogen in peripheral tissues with the help of the aromatase enzyme. Formestane, an aromatase inhibitor, can thus help to decrease the local production of estrogen by blocking the aromatase enzyme in peripheral tissues (ie. Adispose tissue of the breast) to treat hormone sensitive breast cancer.
Female athletes occasionally use clomiphene citrate for the reduction of estrogenicity near the time of a bodybuilding contest. In some instances this may aid in increasing fat loss and muscularity, particularly in female trouble areas such as the hips and thighs. The drug, however, often produces very troubling side effects in pre-menopausal women, and is likewise not in very high demand among this group.
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